. "RIV/60162694:G44__/10:00002402!RIV11-MO0-G44_____" . . . "Holas, Ond\u0159ej" . "CZ - \u010Cesk\u00E1 republika" . . "1210-7816" . "Evaluation of the reactivating efficacy of selected reactivators of paraoxon-inhibited acetylcholinesterase in vitro"@en . . "P(ME09086), S" . "Hodnocen\u00ED reaktiva\u010Dn\u00ED \u00FA\u010Dinnosti vybrann\u00FDch reaktiv\u00E1tor\u016F Paraoxonem inhibovan\u00E9 acetylcholinesterasy in vitro"@cs . "Ku\u010Da, Kamil" . "1" . . . . . . "RIV/60162694:G44__/10:00002402" . "[BB3C6E162C81]" . "59" . "acetylcholinesterase; organophosphorus pesticide; reactivator; in vitro; SAR"@en . "Hodnocen\u00ED reaktiva\u010Dn\u00ED \u00FA\u010Dinnosti vybrann\u00FDch reaktiv\u00E1tor\u016F Paraoxonem inhibovan\u00E9 acetylcholinesterasy in vitro"@cs . "G44" . "Evaluation of the reactivating efficacy of selected reactivators of paraoxon-inhibited acetylcholinesterase in vitro"@en . . "2"^^ . . "5"^^ . . "Hodnocen\u00ED reaktiva\u010Dn\u00ED \u00FA\u010Dinnosti vybrann\u00FDch reaktiv\u00E1tor\u016F Paraoxonem inhibovan\u00E9 acetylcholinesterasy in vitro" . "\u010Cesk\u00E1 a slovensk\u00E1 farmacie" . "4"^^ . . . "Organofosforov\u00E9 pesticidy (OFP) pat\u0159\u00ED do skupiny vysoce toxick\u00FDch ireverzibiln\u00EDch inhibitor\u016F acetylcholinesterase (AChE). Kauz\u00E1ln\u00EDmi l\u00E9\u010Divy p\u0159i intoxikac\u00EDch OFP jsou oximov\u00E9 reaktiv\u00E1tory AChE. Reaktiva\u010Dn\u00ED \u00FA\u010Dinnost 5 nov\u011B p\u0159ipraven\u00FDch bispyridiniov\u00FDch reaktiv\u00E1tor\u016F acetylcholinesterasy byla otestov\u00E1na na modelu paraoxonem inhibovan\u00E9ho enzymu. Reaktiva\u010Dn\u00ED \u00FA\u010Dinnost byla testov\u00E1na za pomoci standardn\u00EDho in vitro testu, kde byl jako zdroj acetylcholinesterasy pou\u017Eit homogen\u00E1t mozku laboratorn\u00EDho potkana. V\u00FDsledky byly porovn\u00E1ny s 5 komer\u010Dn\u011B dostupn\u00FDmi reaktiv\u00E1tory AChE." . "261930" . "The reactivation efficacy of five newly prepared bispyridinium reactivators of acetylcholinesterase was tested on a model of paraoxon-inhibited enzyme. Laboratory rat brain homogenate was used as the source of the AChE. The results were compared with five commercially available AChE reactivators."@en . "Mus\u00EDlek, Kamil" . . . "Opletalov\u00E1, Veronika" . "Organofosforov\u00E9 pesticidy (OFP) pat\u0159\u00ED do skupiny vysoce toxick\u00FDch ireverzibiln\u00EDch inhibitor\u016F acetylcholinesterase (AChE). Kauz\u00E1ln\u00EDmi l\u00E9\u010Divy p\u0159i intoxikac\u00EDch OFP jsou oximov\u00E9 reaktiv\u00E1tory AChE. Reaktiva\u010Dn\u00ED \u00FA\u010Dinnost 5 nov\u011B p\u0159ipraven\u00FDch bispyridiniov\u00FDch reaktiv\u00E1tor\u016F acetylcholinesterasy byla otestov\u00E1na na modelu paraoxonem inhibovan\u00E9ho enzymu. Reaktiva\u010Dn\u00ED \u00FA\u010Dinnost byla testov\u00E1na za pomoci standardn\u00EDho in vitro testu, kde byl jako zdroj acetylcholinesterasy pou\u017Eit homogen\u00E1t mozku laboratorn\u00EDho potkana. V\u00FDsledky byly porovn\u00E1ny s 5 komer\u010Dn\u011B dostupn\u00FDmi reaktiv\u00E1tory AChE."@cs . . "Hodnocen\u00ED reaktiva\u010Dn\u00ED \u00FA\u010Dinnosti vybrann\u00FDch reaktiv\u00E1tor\u016F Paraoxonem inhibovan\u00E9 acetylcholinesterasy in vitro" . .