"V sou\u010Dasnosti vyvinut\u00E9 selektivn\u00ED modul\u00E1tory progesteronov\u00E9ho receptoru (SPRM) jsou steroidn\u00ED slou\u010Deniny s velk\u00FDm substituentem na uhl\u00EDku 11. Interaguj\u00ED s progesteronov\u00FDm receptorem a vykazuj\u00ED antagonistick\u00E9 nebo/a agonistick\u00E9 \u00FA\u010Dinky. Mifepriston byl schv\u00E1len k ukon\u010Den\u00ED gravidity a ulipristalacet\u00E1t jako pohotovostn\u00ED kontracepce a farmakologick\u00E1 l\u00E9\u010Dba d\u011Blo\u017En\u00EDch myom\u016F. SPRM inhibuj\u00ED proliferaci endometria a r\u016Fst myom\u016F a p\u0159edpokl\u00E1d\u00E1 se l\u00E9\u010Debn\u00FD efekt v p\u0159\u00EDpadech endometri\u00F3zy a jin\u00FDch estrogen-dependentn\u00EDch chorob."@cs . . "1" . "RIV/00216208:11110/13:10192340" . . "V\u00FDznam infekc\u00ED zp\u016Fsoben\u00FDch lidsk\u00FDmi papilomaviry" . . . "Currently developed selective progesterone receptor modulators (SPRMs) are steroid derived compounds with a bulky radical substitution at carbon 11. They interact with progesterone receptor and exert antagonistic or/and agonistic effects. Mifepristone was approved for pregnancy termination and ulipristal acetate as emergency contraception and pharmacological therapy of uterine fibroids. SPRMs inhibit endometrial proliferation and myoma growth, this suggests a therapeutical effect in cases of endometriosis and other estrogen-dependent diseases."@en . "[918979E0B9C7]" . . "RIV/00216208:11110/13:10192340!RIV14-MSM-11110___" . . "Selective progesterone receptor modulators and their therapeutical use"@en . . . . "laryngeal papillomatosis; genital warts; esophageal cancer; oropharyngeal cancer; penile cancer; vaginal cancer; vulvar cancer; cervical cancer; human papillomavirus"@en . "Dri\u00E1k, Daniel" . "Selective progesterone receptor modulators and their therapeutical use"@en . . . "152" . "11110" . . "V\u00FDznam infekc\u00ED zp\u016Fsoben\u00FDch lidsk\u00FDmi papilomaviry" . . "http://www.prolekare.cz/casopis-lekaru-ceskych-clanek/vyznam-infekci-zpusobenych-lidskymi-papilomaviry-39863" . . . . . . "V\u00FDznam infekc\u00ED zp\u016Fsoben\u00FDch lidsk\u00FDmi papilomaviry"@cs . "Sehnal, Borek" . "\u010Casopis l\u00E9ka\u0159\u016F \u010Desk\u00FDch" . "116752" . "V" . . "V\u00FDznam infekc\u00ED zp\u016Fsoben\u00FDch lidsk\u00FDmi papilomaviry"@cs . "CZ - \u010Cesk\u00E1 republika" . "V sou\u010Dasnosti vyvinut\u00E9 selektivn\u00ED modul\u00E1tory progesteronov\u00E9ho receptoru (SPRM) jsou steroidn\u00ED slou\u010Deniny s velk\u00FDm substituentem na uhl\u00EDku 11. Interaguj\u00ED s progesteronov\u00FDm receptorem a vykazuj\u00ED antagonistick\u00E9 nebo/a agonistick\u00E9 \u00FA\u010Dinky. Mifepriston byl schv\u00E1len k ukon\u010Den\u00ED gravidity a ulipristalacet\u00E1t jako pohotovostn\u00ED kontracepce a farmakologick\u00E1 l\u00E9\u010Dba d\u011Blo\u017En\u00EDch myom\u016F. SPRM inhibuj\u00ED proliferaci endometria a r\u016Fst myom\u016F a p\u0159edpokl\u00E1d\u00E1 se l\u00E9\u010Debn\u00FD efekt v p\u0159\u00EDpadech endometri\u00F3zy a jin\u00FDch estrogen-dependentn\u00EDch chorob." . "0008-7335" . "2"^^ . "2"^^ . . "5"^^ . . .