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Statements

Subject Item
n2:RIV%2F61389030%3A_____%2F10%3A00352738%21RIV11-GA0-61389030
rdf:type
n13:Vysledek skos:Concept
dcterms:description
L'invention concerne à 3 -, 5 -,7-pyrazolo trisubstitués (4,3-d) pyrimidines représenté par la formule générale (I), et alkyle, cycloalkyle, cyclohétéroalkyle, cycloalkyle, alkyle, aryle ou alkylaryle, R5 est halogène,-NHNH2,-NHOH, NHCONH2, guanylo (NH-C (NH) NH2) éventuellement substitué C1-C6 alkyle, alcényle, alcynyle, cycloalkyle en C3-C15, Rf (cycloalkyle en C3-C15), un hétérocycle, hétéroalkyle, aryle , hétéroaryle, arylalkyle, cyclohétéroalkyle, alkyle cyclohétéroalkyle, hétéroarylalkyle groupe etc.Cette invention concerne de nouveaux pyrazolo (4,3-d) pyrimidine et leur utilisation dans les services publics appropriés, en particulier les méthodes diagnostiques et thérapeutiques. Plus précisément, la présente invention concerne également l'utilisation du 3,5,7-pyrazolo trisubstitués (4,3-d) pyrimidines ou un sel pharmaceutiquement acceptable de celui-ci en combinaison avec des cytostatiques dans la préparation d'un médicament pour traiter le cancer. The invention relates to 3-,5-,7-trisubstituted pyrazolo(4,3-d)pyrimidines represented by the general formula (I), and substituted alkyl, cycloalkyl, cycloheteroalkyl, cycloalkyl, alkyl, aryl or alkylaryl group, R5 is halogen, -NHNH2, -NHOH, NHCONH2, guanylo (NH-C(NH)NH2) an optionally substituted C1-C6 alkyl, alkenyl, alkinyl, C3-C15 cycloalkyl, Rf (C3-C15 cycloalkyl), heterocycle, heteroalkyl, aryl, heteroaryl, arylalkyl, cycloheteroalkyl, cycloheteroalkyl alkyl, heteroarylalkyl group etc.This invention relates to new pyrazolo(4,3-d)pyrimidine derivatives and to their use in suitable utilities, especially diagnostic and therapeutic methods. More specifically, the present invention also relates to the use of 3,5,7-trisubstituted pyrazolo(4,3-d)pyrimidines or a pharmaceutically acceptable salt thereof in combination with cytostatics in the preparation of a medicament for treating cancer.
dcterms:title
Nouveaux pyrazolo[4,3-D]pyrimidines, procedes pour leur preparation et methodes Novel pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy
skos:prefLabel
Novel pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy Nouveaux pyrazolo[4,3-D]pyrimidines, procedes pour leur preparation et methodes
skos:notation
RIV/61389030:_____/10:00352738!RIV11-GA0-61389030
n3:aktivita
n16:P
n3:aktivity
P(GA301/08/1649), P(GA522/09/1576)
n3:cisloPatentuVzoru
CA2480409
n3:datumUdeleniPatentuVzoru
2010-06-22+02:00
n3:dodaniDat
n14:2011
n3:domaciTvurceVysledku
n5:4712048 n5:9896821 n5:9961216 n5:9130241 n5:1870378
n3:druhVysledku
n15:P
n3:duvernostUdaju
n9:S
n3:entitaPredkladatele
n17:predkladatel
n3:idSjednocenehoVysledku
275179
n3:idVysledku
RIV/61389030:_____/10:00352738
n3:jazykVysledku
n19:fre
n3:klicovaSlova
novel pyrazolo[4,3-D]pyrimidines; process; preparation; method; therapy
n3:klicoveSlovo
n8:novel%20pyrazolo%5B4 n8:preparation n8:3-D%5Dpyrimidines n8:therapy n8:process n8:method
n3:kontrolniKodProRIV
[07A1E6EA1DC4]
n3:licencniPoplatek
n4:A
n3:mistoVydaniPatentuVzoru
Ottawa
n3:nazevVydavatelePatentuVzoru
Canadian Intellectual Property Office http://brevets-patents.ic.gc.ca/opic-cipo/cpd/eng/patent/2480409/summary.html?type=number_search
n3:obor
n10:FD
n3:pocetDomacichTvurcuVysledku
5
n3:pocetTvurcuVysledku
5
n3:projekt
n20:GA301%2F08%2F1649 n20:GA522%2F09%2F1576
n3:rokUplatneniVysledku
n14:2010
n3:statVydaniPatentuVzoru
n11:CA
n3:tvurceVysledku
Lenobel, René Kryštof, Vladimír Havlíček, Libor Moravcová, Daniela Strnad, Miroslav
n3:uzemniOchranaPatentu
n21:D
n3:vlastnik
n17:vlastnikVysledku
n3:vyuzitiJinymSubjektem
n7:A
n3:vyuzitiPatentuVzoru
n18:B
n3:vlastnikPatentuVzoru
Ústav experimentální botaniky AV ČR, v. v. i., Univerzita Palackého v Olomouci