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rdf:type
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Description
| - 20-oxo-5beta-pregnan-3alpha-yl sulfát (3alfa5betaS) je inhibitor NMDA receptorů, jehož působení závisí na aktivaci NMDA receptorů. 3alfa5betaS inhibuje iontové kanály NMDA receptorů snižováním pravděpodobnosti jejich otevírání. Inhibiční účinky 3alfa5betaS jsou menší u proudových odpovědí NMDA receptorů, které jsou aktivované glutamátem uvolněným během synaptického přenosu, než receptorů aktivovaných tonicky (cs)
- 20-oxo-5beta-pregnan-3alpha-yl sulfate (3alfa5betaS) is a use-dependent but voltage-independent inhibitor of NMDA receptors that exerts its effect by reducing the peak Po of NMDA receptor channels. Its inhibitory action is weaker for responses mediated by NMDA receptors activated by synaptically released glutamate than those tonically activated by the agonist
- 20-oxo-5beta-pregnan-3alpha-yl sulfate (3alfa5betaS) is a use-dependent but voltage-independent inhibitor of NMDA receptors that exerts its effect by reducing the peak Po of NMDA receptor channels. Its inhibitory action is weaker for responses mediated by NMDA receptors activated by synaptically released glutamate than those tonically activated by the agonist (en)
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Title
| - 20-oxo-5beta-pregnan-3alpha-yl sulfate is a use-dependent NMDA receptor inhibitor
- 20-oxo-5beta-pregnan-3alpha-yl sulfate is a use-dependent NMDA receptor inhibitor (en)
- 20-oxo-5beta-pregnan-3alpha-yl sulfát je inhibitor NMDA receptorů závislý na jejich aktivaci (cs)
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skos:prefLabel
| - 20-oxo-5beta-pregnan-3alpha-yl sulfate is a use-dependent NMDA receptor inhibitor
- 20-oxo-5beta-pregnan-3alpha-yl sulfate is a use-dependent NMDA receptor inhibitor (en)
- 20-oxo-5beta-pregnan-3alpha-yl sulfát je inhibitor NMDA receptorů závislý na jejich aktivaci (cs)
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skos:notation
| - RIV/67985823:_____/05:00024112!RIV06-AV0-67985823
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http://linked.open.../vavai/riv/strany
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http://linked.open...avai/riv/aktivita
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http://linked.open...avai/riv/aktivity
| - P(1M0517), P(GA309/04/1537), P(LC554), Z(AV0Z50110509)
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http://linked.open...iv/cisloPeriodika
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http://linked.open...vai/riv/dodaniDat
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http://linked.open...aciTvurceVysledku
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http://linked.open.../riv/druhVysledku
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http://linked.open...iv/duvernostUdaju
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http://linked.open...titaPredkladatele
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http://linked.open...dnocenehoVysledku
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http://linked.open...ai/riv/idVysledku
| - RIV/67985823:_____/05:00024112
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http://linked.open...riv/jazykVysledku
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http://linked.open.../riv/klicovaSlova
| - neurosteroids; NMDA receptor; inhibition (en)
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http://linked.open.../riv/klicoveSlovo
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http://linked.open...odStatuVydavatele
| - US - Spojené státy americké
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http://linked.open...ontrolniKodProRIV
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http://linked.open...i/riv/nazevZdroje
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http://linked.open...in/vavai/riv/obor
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http://linked.open...ichTvurcuVysledku
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http://linked.open...cetTvurcuVysledku
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http://linked.open...vavai/riv/projekt
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http://linked.open...UplatneniVysledku
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http://linked.open...v/svazekPeriodika
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http://linked.open...iv/tvurceVysledku
| - Chodounská, Hana
- Horák, Martin
- Vyklický ml., Ladislav
- Petrovič, Miloš
- Sedláček, Miloslav
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http://linked.open...n/vavai/riv/zamer
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issn
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number of pages
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is http://linked.open...avai/riv/vysledek
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