Byla syntetizována skupina nových derivátů N-benzylsalicylthioamidů; sloučeniny byly testovány in vitro na antimykobakteriální aktivitu proti Mycobacterium tuberculosis, Mycobacterium kansasii a Mycobacterium avium; pro hodnocení vztahu struktura-účinek byl použit Topplissův postup (cs)
The group of new derivatives of N-benzylsalicylthioamides was synthesized and the compounds were tested for in vitro antimycobacterial activity against Mycobacterium tuberculosis, Mycobacterium kansasii and Mycobacterium avium; Toppliss approach was used for the SAR study
The group of new derivatives of N-benzylsalicylthioamides was synthesized and the compounds were tested for in vitro antimycobacterial activity against Mycobacterium tuberculosis, Mycobacterium kansasii and Mycobacterium avium; Toppliss approach was used for the SAR study (en)