About: Inhibitory effects of memantine on human cytochrome P450 activities: prediction of in vivo drug interactions     Goto   Sponge   NotDistinct   Permalink

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Description
  • The aim of the present study was to predict the drug interaction potential of memantine by elucidation of its inhibitory effects on cytochrome P450 enzymes using pooled human liver microsomes (HLM) and recombinant P450s.
  • The aim of the present study was to predict the drug interaction potential of memantine by elucidation of its inhibitory effects on cytochrome P450 enzymes using pooled human liver microsomes (HLM) and recombinant P450s. (en)
  • Cílem prezentované studie bylo hodnocení potenciálních lékových interakcí memantinu, a to hodnocením jeho inhibičního vlivu na aktivity cytochromů P450 za použití lidských jaterních mikrozomů a rekombinantních enzymů. (cs)
Title
  • Inhibitory effects of memantine on human cytochrome P450 activities: prediction of in vivo drug interactions
  • Inhibitory effects of memantine on human cytochrome P450 activities: prediction of in vivo drug interactions (en)
  • Inhibiční vliv memantinu na aktivitu lidských cytochromů P450: predikce in vivo lékových interakcí (cs)
skos:prefLabel
  • Inhibitory effects of memantine on human cytochrome P450 activities: prediction of in vivo drug interactions
  • Inhibitory effects of memantine on human cytochrome P450 activities: prediction of in vivo drug interactions (en)
  • Inhibiční vliv memantinu na aktivitu lidských cytochromů P450: predikce in vivo lékových interakcí (cs)
skos:notation
  • RIV/00216208:11150/04:00002063!RIV/2005/MSM/111505/N
http://linked.open.../vavai/riv/strany
  • 583;589
http://linked.open...avai/riv/aktivita
http://linked.open...avai/riv/aktivity
  • P(OC B15.30)
http://linked.open...iv/cisloPeriodika
  • 8
http://linked.open...vai/riv/dodaniDat
http://linked.open...aciTvurceVysledku
http://linked.open.../riv/druhVysledku
http://linked.open...iv/duvernostUdaju
http://linked.open...titaPredkladatele
http://linked.open...dnocenehoVysledku
  • 568234
http://linked.open...ai/riv/idVysledku
  • RIV/00216208:11150/04:00002063
http://linked.open...riv/jazykVysledku
http://linked.open.../riv/klicovaSlova
  • memantine; cytochrome P450 2B6; selective inhibition (en)
http://linked.open.../riv/klicoveSlovo
http://linked.open...odStatuVydavatele
  • DE - Spolková republika Německo
http://linked.open...ontrolniKodProRIV
  • [48E5A30D2875]
http://linked.open...i/riv/nazevZdroje
  • European Journal of Clinical Pharmacology
http://linked.open...in/vavai/riv/obor
http://linked.open...ichTvurcuVysledku
http://linked.open...cetTvurcuVysledku
http://linked.open...vavai/riv/projekt
http://linked.open...UplatneniVysledku
http://linked.open...v/svazekPeriodika
  • 60
http://linked.open...iv/tvurceVysledku
  • Chládek, Jaroslav
  • Mičuda, Stanislav
  • Martínková, Jiřina
  • Mundlová, Lucie
issn
  • 0031-6970
number of pages
http://localhost/t...ganizacniJednotka
  • 11150
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