About: In vitro expression of recombinant protein CYP3A4 for study of metabolic changes of drugs:feasibility study     Goto   Sponge   NotDistinct   Permalink

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Description
  • The project is focussed on feasibility study of recombinant expression of CYP3A4 enzyme for in virto tests of drug biotransformation. The project is based on cloning gene for CYP3A4 into baculovirus expression vector and succesive production of the enzyme in insect host cells in vitro. (en)
  • Projekt je zaměřen na studium proveditelnosti rekombinantní systémy enzymu CYP3A4 pro použití k in vitro studiu biotransformace léčiv. Projekt je založen na inkorporaci genu pro CYP3A4 do bakulovirového expresního vektoru a produkci enzymu ve hmyzích hostitelských buňkách in vitro.
Title
  • In vitro expression of recombinant protein CYP3A4 for study of metabolic changes of drugs:feasibility study (en)
  • In vitro exprese rekombinantního proteinu CYP3A4 pro studium metabolických přeměn léčiv: studium proveditelnosti
skos:notation
  • NL6177
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  • CYP3A4;vector;feasibility;recombinant;baculovirus;biotransformation;molecular;drug (en)
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  • Cílem projektu bylo vypracovat metodu rekombinantní syntézy cytochromu P450 3A4, jeho inkorporace do vektoru až po následnou produkci enzymu v hmyzích buňkách. Zvládnutí moderních metod. (cs)
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  • feasibility
  • baculovirus
  • biotransformation
  • vector
  • recombinant
  • molecular
  • CYP3A4
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