About: Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone     Goto   Sponge   NotDistinct   Permalink

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Description
  • Amiodarone, an ion channel blocker in clinical use as an antiarrhythmic agent, exhibits broad range fungicidal effects. We show that a polarized membrane is critical for drug toxicity; furthermore, the change in membrane potential precedes and is closely coupled to both cation influx and cell death
  • Amiodarone, an ion channel blocker in clinical use as an antiarrhythmic agent, exhibits broad range fungicidal effects. We show that a polarized membrane is critical for drug toxicity; furthermore, the change in membrane potential precedes and is closely coupled to both cation influx and cell death (en)
  • Amiodaron, blokátor iontových kanálů, který se v klinické praxi používá pro léčbu srdečních arytmií, má zároveň širokospektré antifungální účinky. Práce ukazuje, že jeho toxické účinky jsou podmíněny elektrochemickým potenciálem na membráně a že změna membránového potenciálu předchází vniku kationtů a buněčné smrti (cs)
Title
  • Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone
  • Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone (en)
  • Hyperpolarizace membrány je příčinou vniku kationtů a antifungální aktivity amiodaronu (cs)
skos:prefLabel
  • Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone
  • Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone (en)
  • Hyperpolarizace membrány je příčinou vniku kationtů a antifungální aktivity amiodaronu (cs)
skos:notation
  • RIV/67985823:_____/09:00323535!RIV09-AV0-67985823
http://linked.open...avai/riv/aktivita
http://linked.open...avai/riv/aktivity
  • P(KJB500110701), P(LC531), Z(AV0Z50110509)
http://linked.open...iv/cisloPeriodika
  • 5
http://linked.open...vai/riv/dodaniDat
http://linked.open...aciTvurceVysledku
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http://linked.open...iv/duvernostUdaju
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http://linked.open...dnocenehoVysledku
  • 325301
http://linked.open...ai/riv/idVysledku
  • RIV/67985823:_____/09:00323535
http://linked.open...riv/jazykVysledku
http://linked.open.../riv/klicovaSlova
  • membrane potential; S. cerevisiae; cation fluxes (en)
http://linked.open.../riv/klicoveSlovo
http://linked.open...odStatuVydavatele
  • US - Spojené státy americké
http://linked.open...ontrolniKodProRIV
  • [A8997D4443E2]
http://linked.open...i/riv/nazevZdroje
  • Journal of Biological Chemistry
http://linked.open...in/vavai/riv/obor
http://linked.open...ichTvurcuVysledku
http://linked.open...cetTvurcuVysledku
http://linked.open...vavai/riv/projekt
http://linked.open...UplatneniVysledku
http://linked.open...v/svazekPeriodika
  • 284
http://linked.open...iv/tvurceVysledku
  • Marešová, Lydie
  • Sychrová, Hana
  • Muend, S.
  • Rao, R.
  • Zhang, Y. Q.
http://linked.open...ain/vavai/riv/wos
  • 262700900022
http://linked.open...n/vavai/riv/zamer
issn
  • 0021-9258
number of pages
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