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Description
  • Metodou terčíkového zámku (patch-clamp) byly studovány účinky physostigminu na myší svalové nikotinické acetylcholinové receptory exprimované v linii COS–7 buněk. Physostigmin alosterickým mechanismem urychloval desentizaci a snižoval velikost proudů vyvolaných aplikací acetylcholinu (cs)
  • The action of physostigmine on mouse nicotinic acetylcholine receptor expressed in the COS–7 cell line was studiem by the patch-clamp technique. Physostigmine accelerated, by allosteric modulation, the rat of desensitization of whole cell currents induced by acetylcholine and decreased the maximal amplitude in concentration-dependent manner
  • The action of physostigmine on mouse nicotinic acetylcholine receptor expressed in the COS–7 cell line was studiem by the patch-clamp technique. Physostigmine accelerated, by allosteric modulation, the rat of desensitization of whole cell currents induced by acetylcholine and decreased the maximal amplitude in concentration-dependent manner (en)
Title
  • Allosteric modulation of the nicotinic acetylcholine receptor by physostigmine
  • Alosterická modulace nikotinického acetylcholinového receptoru physostigminem (cs)
  • Allosteric modulation of the nicotinic acetylcholine receptor by physostigmine (en)
skos:prefLabel
  • Allosteric modulation of the nicotinic acetylcholine receptor by physostigmine
  • Alosterická modulace nikotinického acetylcholinového receptoru physostigminem (cs)
  • Allosteric modulation of the nicotinic acetylcholine receptor by physostigmine (en)
skos:notation
  • RIV/67985823:_____/05:00024057!RIV06-AV0-67985823
http://linked.open.../vavai/riv/strany
  • 355;358
http://linked.open...avai/riv/aktivita
http://linked.open...avai/riv/aktivity
  • P(GA202/02/1213), P(GA305/02/1333), P(GD305/03/H148), Z(AV0Z5011922)
http://linked.open...iv/cisloPeriodika
  • -
http://linked.open...vai/riv/dodaniDat
http://linked.open...aciTvurceVysledku
http://linked.open.../riv/druhVysledku
http://linked.open...iv/duvernostUdaju
http://linked.open...titaPredkladatele
http://linked.open...dnocenehoVysledku
  • 511747
http://linked.open...ai/riv/idVysledku
  • RIV/67985823:_____/05:00024057
http://linked.open...riv/jazykVysledku
http://linked.open.../riv/klicovaSlova
  • nicotinic ACh receptor; serine; desensitization (en)
http://linked.open.../riv/klicoveSlovo
http://linked.open...odStatuVydavatele
  • US - Spojené státy americké
http://linked.open...ontrolniKodProRIV
  • [F855E316C414]
http://linked.open...i/riv/nazevZdroje
  • New York Academy of Sciences. Annals
http://linked.open...in/vavai/riv/obor
http://linked.open...ichTvurcuVysledku
http://linked.open...cetTvurcuVysledku
http://linked.open...vavai/riv/projekt
http://linked.open...UplatneniVysledku
http://linked.open...v/svazekPeriodika
  • 1048
http://linked.open...iv/tvurceVysledku
  • Vyskočil, František
  • Krůšek, Jan
  • Svobodová, Lucie
  • Hendrych, Tomáš
http://linked.open...n/vavai/riv/zamer
issn
  • 0077-8923
number of pages
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