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rdf:type
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Description
| - A number of structurally diverse nucleosides phosphonic acids have been tested against human recombinant thymidine phosphorylase and human platelets supernatant using 2'-deoxy-5-nitrouridine as the substrate. We have selected several inhibitors working at micromolar level as lead structures for further evaluation.
- A number of structurally diverse nucleosides phosphonic acids have been tested against human recombinant thymidine phosphorylase and human platelets supernatant using 2'-deoxy-5-nitrouridine as the substrate. We have selected several inhibitors working at micromolar level as lead structures for further evaluation. (en)
- Řada strukturně odlišných nukleosidfosfonových kyselin byla testována v interakci s rekombinantní thymidinfosforylázou a supernatantem lidských krevních destiček za užití 2'-deoxy-5-nitrouridinu jako substrátu. Bylo nalezeno několik inhibitorů působících na mikromolární úrovni jakožto klíčové struktury pro další studium. (cs)
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Title
| - Nucleoside phosphonic acids in thymidine phosphorylase inhibition: Structure - activity relationship
- Nukleosidfosfonové kyseliny jako inhibitory thymidinfosforylázy: vztah struktury a aktivity (cs)
- Nucleoside phosphonic acids in thymidine phosphorylase inhibition: Structure - activity relationship (en)
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skos:prefLabel
| - Nucleoside phosphonic acids in thymidine phosphorylase inhibition: Structure - activity relationship
- Nukleosidfosfonové kyseliny jako inhibitory thymidinfosforylázy: vztah struktury a aktivity (cs)
- Nucleoside phosphonic acids in thymidine phosphorylase inhibition: Structure - activity relationship (en)
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skos:notation
| - RIV/61388963:_____/08:00312445!RIV09-AV0-61388963
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http://linked.open...avai/riv/aktivita
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http://linked.open...avai/riv/aktivity
| - P(LC06061), P(LC06077), P(LC512), Z(AV0Z40550506)
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http://linked.open...iv/cisloPeriodika
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http://linked.open...vai/riv/dodaniDat
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http://linked.open...aciTvurceVysledku
| - Pačes, Ondřej
- Kočalka, Petr
- Rosenberg, Ivan
- Petrová, Magdalena
- Rejman, Dominik
- Kovačková, Soňa
- Točík, Zdeněk
- Kóšiová, Ivana
- Králíková, Šárka
- Páv, Ondřej
- Liboska, Radek
- Vaněk, Václav
- Panova, Natalya
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http://linked.open.../riv/druhVysledku
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http://linked.open...iv/duvernostUdaju
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http://linked.open...titaPredkladatele
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http://linked.open...dnocenehoVysledku
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http://linked.open...ai/riv/idVysledku
| - RIV/61388963:_____/08:00312445
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http://linked.open...riv/jazykVysledku
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http://linked.open.../riv/klicovaSlova
| - thymidine phosphorylase; inhibitors; phosphonic acids (en)
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http://linked.open.../riv/klicoveSlovo
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http://linked.open...odStatuVydavatele
| - GB - Spojené království Velké Británie a Severního Irska
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http://linked.open...ontrolniKodProRIV
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http://linked.open...i/riv/nazevZdroje
| - Nucleic Acids Symposium Series
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http://linked.open...in/vavai/riv/obor
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http://linked.open...ichTvurcuVysledku
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http://linked.open...cetTvurcuVysledku
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http://linked.open...vavai/riv/projekt
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http://linked.open...UplatneniVysledku
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http://linked.open...v/svazekPeriodika
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http://linked.open...iv/tvurceVysledku
| - Petrová, Magdalena
- Rosenberg, Ivan
- Vaněk, Václav
- Kovačková, Soňa
- Rejman, Dominik
- Králíková, Šárka
- Kóšiová, Ivana
- Panova, Natalya
- Páv, Ondřej
- Točík, Zdeněk
- Liboska, Radek
- Kočalka, Petr
- Pačes, Ondřej
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http://linked.open...n/vavai/riv/zamer
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issn
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number of pages
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