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Description
| - Series of ten N-substituted 2-(aminoethyl)-6-fluorobenzothiazoles inhibited photosynthetic electron transport in spinach chloroplasts. The inhibitory activity linearly increased with hydrophobic contributions (expressed as hydrophobic constants pi) and molar volumes of individual substituents in C-(2) position of 6-fluorobenzothiazole scaffold to the optima pi ca. 2 and MV ca. 233 cm(3), while for more lipophilic and/or bulkier derivatives PET inhibiting activity linearly decreased. The site of inhibitory action of the tested compounds is situated on the donor side of photosystem II, and interaction of these compounds with aromatic amino acid residues in photosynthetic proteins was confirmed by fluorescence spectroscopy. Synthesis and characterization of five new N alpha-(alkoxycarbonyl)-N-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-l-phenylalaninamides is presented as well.
- Series of ten N-substituted 2-(aminoethyl)-6-fluorobenzothiazoles inhibited photosynthetic electron transport in spinach chloroplasts. The inhibitory activity linearly increased with hydrophobic contributions (expressed as hydrophobic constants pi) and molar volumes of individual substituents in C-(2) position of 6-fluorobenzothiazole scaffold to the optima pi ca. 2 and MV ca. 233 cm(3), while for more lipophilic and/or bulkier derivatives PET inhibiting activity linearly decreased. The site of inhibitory action of the tested compounds is situated on the donor side of photosystem II, and interaction of these compounds with aromatic amino acid residues in photosynthetic proteins was confirmed by fluorescence spectroscopy. Synthesis and characterization of five new N alpha-(alkoxycarbonyl)-N-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-l-phenylalaninamides is presented as well. (en)
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Title
| - Synthesis and photosynthetic electron transport inhibition of 2-substituted 6-fluorobenzothiazoles
- Synthesis and photosynthetic electron transport inhibition of 2-substituted 6-fluorobenzothiazoles (en)
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skos:prefLabel
| - Synthesis and photosynthetic electron transport inhibition of 2-substituted 6-fluorobenzothiazoles
- Synthesis and photosynthetic electron transport inhibition of 2-substituted 6-fluorobenzothiazoles (en)
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skos:notation
| - RIV/62157124:16370/14:43872711!RIV15-MSM-16370___
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http://linked.open...avai/riv/aktivita
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http://linked.open...avai/riv/aktivity
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http://linked.open...iv/cisloPeriodika
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http://linked.open...vai/riv/dodaniDat
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http://linked.open...aciTvurceVysledku
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http://linked.open.../riv/druhVysledku
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http://linked.open...iv/duvernostUdaju
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http://linked.open...titaPredkladatele
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http://linked.open...dnocenehoVysledku
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http://linked.open...ai/riv/idVysledku
| - RIV/62157124:16370/14:43872711
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http://linked.open...riv/jazykVysledku
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http://linked.open.../riv/klicovaSlova
| - Structure-activity relationships; Bioorganic chemistry; Herbicidal activity; Photosynthetic electron transport; Heterocycles (en)
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http://linked.open.../riv/klicoveSlovo
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http://linked.open...odStatuVydavatele
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http://linked.open...ontrolniKodProRIV
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http://linked.open...i/riv/nazevZdroje
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http://linked.open...in/vavai/riv/obor
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http://linked.open...ichTvurcuVysledku
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http://linked.open...cetTvurcuVysledku
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http://linked.open...UplatneniVysledku
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http://linked.open...v/svazekPeriodika
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http://linked.open...iv/tvurceVysledku
| - Jampílek, Josef
- Imramovský, Aleš
- Kráľová, Katarína
- Peško, Matúš
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http://linked.open...ain/vavai/riv/wos
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issn
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number of pages
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http://bibframe.org/vocab/doi
| - 10.1007/s00706-014-1283-9
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http://localhost/t...ganizacniJednotka
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