About: A-204C polymorphism and regulation of cholesterol 7alpha-hydroxylase activity     Goto   Sponge   NotDistinct   Permalink

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  • Circadian variation in cholesterol 7alpha-hydroxylase (CYP7A1) activity will be studied in healthy volunteers homozygous either for -204A or -204C variant in CYP7A1 gene promoter. Circadian variation in CYP7A1 activity will be studied under basal conditions and after stimulation and inhibition of CYP7A1 gene expression using drugs (colestipol and chenodeoxycholic acid, respectively). The activity of both CYP7A1 gene promoter variants will be studied in vitro using dual lucipherase assay both under basal conditions and after stimulation. (en)
  • Cirkadiánní variace v aktivitě cholesterol 7alfa-hydroxylázy (CYP7A1) bude studována u zdravých dobrovolníků homozygotních pro variantu -204A nebo -204C v promotoru genu pro CYP7A1. Cirkadiánní variace v aktivitě CYP7A1 bude studována za bazálních podmínek a po stimulaci nebo inhibici exprese genu pro CYP7A1 pomocí léků (colestipolu a kyseliny chenodeoxycholové). Aktivita obou variant promotoru genu pro CYP7A1 bude studována in vitro technikou duální luciferázové eseje jak za bazálních podmínek, tak po stimulaci. (cs)
Title
  • Polymorfismus A-204C a regulace aktivity cholesterol 7alfa-hydroxylázy (cs)
  • A-204C polymorphism and regulation of cholesterol 7alpha-hydroxylase activity (en)
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  • CYP7A1; LDL-cholesterol; circadian variation; genetics; reporter assay (en)
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