About: Anti-inflammatory activity of Macleaya cordata extract and its component in vitro and in vivo     Goto   Sponge   NotDistinct   Permalink

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  • Aerial part of M. cordata is used in Chinese herbal medicine for the treatment of acute or chronic colitis. Quaternary benzofenathridine alkaloids sanguinarine and chelerythrine, the active principle of M. cordata, display a large number of in vitro biological activities (e.g. antimicrobial, anti-inflammatory)and are intensively studied, contrary to protopine and allocryptopine which are also present in M.c. extract, but the informations about their biological activity are rare. The aim of the project is to assess the chemoprotective and/or anti-inflammatory activity of M.c. extract and its main components protopine and allocryptopine in vitro and in vivo in comparison with sanguinarine and chelerythrine. (en)
  • In vitro prokázat protizánětlivý účinek sanguinarinu, chelerythrinu, protopinu a allokryptopinu na signální dráhy spojené s NF-kappaB a Nrf2 v buněčné linii Caco-2. In vivo prokázat účinek alkaloidů na dextransulfátem indukovanou kolitidu u potkana (cs)
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  • Anti-inflammatory activity of Macleaya cordata extract and its component in vitro and in vivo (en)
  • Protizánětlivá aktivita extraktu z Macleaya cordata a jeho hlavních složek in vitro a in vivo (cs)
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  • sanguinarine; chelerythrine; protopine; allocryptopine; dextran sulphate; Caco-2 cells; Macleaya cordata (en)
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